About the Cover: Interaction =
of the β-L-enantiomer of a 4'-C-e=
thynyl-2',3'-dideoxynucleoside analogue (ent-14-TP)=
at the active site of HIV reverse transcriptase (Siddiqui, M. A.; et al=
. J. Med. Chem.2004, 47, 5041-5048).
Han-Cheng Z=
hang, Claudia K. Derian, David F. McComsey, Kimberly B. White, Hong Ye, =
Leonard R. Hecker, Jian Li, Michael F. Addo, Diane Croll, Annette J. Eck=
ardt, Charles E. Smith, Quan Li, Wai-Man Cheung, Bruce R. Conway, Stuart=
Emanuel, Keith T. Demarest, Patricia Andrade-Gordon, Bruce P. Damiano, =
and Bruce E. Maryanoff
pp 1725–1728
Publication D=
ate (Web): November 13, 2004 (Letter)=
span>
Mimi L. Quan, Patrick Y. S=
. Lam, Qi Han, Donald J. P. Pinto, Ming Y. He, Renhua Li, Christopher D.=
Ellis, Charles G. Clark, Christopher A. Teleha, Jung-Hui Sun, Richard S=
. Alexander, Steve Bai, Joseph M. Luettgen, Robert M. Knabb, Pancras C. =
Wong, and Ruth R. Wexler
Pieter Van =
der Veken, Kristel Senten, István Kertèsz, Ingrid De Meest=
er, Anne-Marie Lambeir, Marie-Berthe Maes, Simon Scharpé, Achiel =
Haemers, and Koen Augustyns
pp 1768–1780
Publicat=
ion Date (Web): August 26, 2004 (Articl=
e)
Jörg Holenz, R=
amon Mercè, José Luis Díaz, Xavier Guitart, Xavier =
Codony, Alberto Dordal, Gonzalo Romero, Antoni Torrens, Josep Mas, Blas =
Andaluz, Susana Hernández, Xavier Monroy, Elisabeth Sánche=
z, Enrique Hernández, Raquel Pérez, Roger Cubí, Olg=
a Sanfeliu, and Helmut Buschmann
pp 1781–1795
Pub=
lication Date (Web): September 04, 2004=
(Article)
Sarah Ulmschneider, Ursula Müller-Vieira, Markus M=
itrenga, Rolf W. Hartmann, Sandrine Oberwinkler-Marchais, Christian D. K=
lein, Matthias Bureik, Rita Bernhardt, Iris Antes, and Thomas Lengauer=
div>pp 1796–1805
Publication Date (Web): Augu=
st 27, 2004 (Article)
Dominique L. N. G. Sur=
leraux, Abdellah Tahri, Wim G. Verschueren, Geert M. E. Pille, Herman A.=
de Kock, Tim H. M. Jonckers, Anik Peeters, Sandra De Meyer, Hilde Azijn=
, Rudi Pauwels, Marie-Pierre de Bethune, Nancy M. King, Moses Prabu-Jeya=
balan, Celia A. Schiffer, and Piet B. T. P. Wigerinck
pp 1813&ndash=
;1822
Publication Date (Web): October 05, 2004 (Article)
Jos H. M. Lange, Herman H. van Stuivenberg, Hein K. A. =
C. Coolen, Tiny J. P. Adolfs, Andrew C. McCreary, Hiskias G. Keizer, Hen=
ri C. Wals, Willem Veerman, Alice J. M. Borst, Wouter de Looff, Peter C.=
Verveer, and Chris G. Kruse
pp 1823–1838
Publica=
tion Date (Web): September 29, 2004 (Ar=
ticle)
<=
a href=3D"/doi/abs/10.1021/jm049614v">Discovery of a Potent, Selective, =
and Efficacious Class of Reversible α-Ketoheterocycle Inhibitors =
of Fatty Acid Amide Hydrolase Effective as Analgesics
Dale L. Boger, Hiroshi Miyauchi, Wu Du, Christophe H=
ardouin, Robert A. Fecik, Heng Cheng, Inkyu Hwang, Michael P. Hedrick, D=
onmienne Leung, Orlando Acevedo, Cristiano R. W. Guimarães, Willi=
am L. Jorgensen, and Benjamin F. Cravatt
pp 1849–1856
Publication Date (Web): October 23, 2004 (Article)
Devin M. Swanson, Adrienne E. Dubin, Chandra Shah, Nadia Nasse=
r, Leon Chang, Scott L. Dax, Michele Jetter, J. Guy Breitenbucher, Chang=
lu Liu, Curt Mazur, Brian Lord, Lisa Gonzales, Kenway Hoey, Michele Rizz=
olio, Michael Bogenstaetter, Ellen E. Codd, Doo H. Lee, Sui-Po Zhang, Sa=
ndra R. Chaplan, and Nicholas I. Carruthers
pp 1857–1872
=
Publication Date (Web): November 12, 2004 (Article)
Kristen L. Arienti, Anders Brunmar=
k, Frank U. Axe, Kelly McClure, Alice Lee, Jon Blevitt, Danielle K. Neff=
, Liming Huang, Shelby Crawford, Chennagiri R. Pandit, Lars Karlsson, an=
d J. Guy Breitenbucher
pp 1873–1885
Publication D=
ate (Web): November 05, 2004 (Article)<=
/span>
Gee-Ho=
ng Kuo, Aihua Wang, Stuart Emanuel, Alan DeAngelis, Rui Zhang, Peter J. =
Connolly, William V. Murray, Robert H. Gruninger, Jan Sechler, Angel Fue=
ntes-Pesquera, Dana Johnson, Steven A. Middleton, Linda Jolliffe, and Xi=
n Chen
pp 1886–1900
Publication Date (Web): November 06, 2004 (Article)
Paul A. J. Jansse=
n, Paul J. Lewi, Eddy Arnold, Frits Daeyaert, Marc de Jonge, Jan Heeres,=
Luc Koymans, Maarten Vinkers, Jérôme Guillemont, Elisabeth=
Pasquier, Mike Kukla, Don Ludovici, Koen Andries, Marie-Pierre de B&eac=
ute;thune, Rudi Pauwels, Kalyan Das, Art D. Clark, Jr., Yulia Volovik Fr=
enkel, Stephen H. Hughes, Bart Medaer, Fons De Knaep, Hilde Bohets, Fred=
De Clerck, Ann Lampo, Peter Williams, and Paul Stoffels
pp 1901&nd=
ash;1909
Publication Date (Web): November 06, 2004<=
span class=3D"manType"> (Article)
Jan Heeres, Marc R. de Jonge, Lucien M. H. Koymans,=
Frits F. D. Daeyaert, Maarten Vinkers, Koen J. A. Van Aken, Eddy Arnold=
, Kalyan Das, Amuri Kilonda, Georges J. Hoornaert, Frans Compernolle, Ma=
rek Cegla, Rasha A. Azzam, Koen Andries, Marie-Pierre de Béthune,=
Hilde Azijn, Rudi Pauwels, Paul J. Lewi, and Paul A. J. Janssen
pp=
1910–1918
Publication Date (Web): November 0=
9, 2004 (Article)
Giuseppe Campiani, Caterina Fattorusso, St=
efania Butini, Alessandra Gaeta, Marianna Agnusdei, Sandra Gemma, Marco =
Persico, Bruno Catalanotti, Luisa Savini, Vito Nacci, Ettore Novellino, =
Harold W. Holloway, Nigel H. Greig, Tatyana Belinskaya, James M. Fedorko=
, and Ashima Saxena
pp 1919–1929
Publication Date=
(Web): November 16, 2004 (Article)
Dominique L. N. G. Sur=
leraux, Herman A. de Kock, Wim G. Verschueren, Geert M. E. Pille, Louis =
J. R. Maes, Anik Peeters, Sandrine Vendeville, Sandra De Meyer, Hilde Az=
ijn, Rudi Pauwels, Marie-Pierre de Bethune, Nancy M. King, Moses Prabu-J=
eyabalan, Celia A. Schiffer, and Piet B. T. P. Wigerinck
pp 1965&nd=
ash;1973
Publication Date (Web): January 25, 2005 (Article)
Chi B. Vu, Deborah Pan, Bo Peng, Gnanasambandam Kumaravel, Glen=
n Smits, Xiaowei Jin, Deepali Phadke, Thomas Engber, Carol Huang, Jennif=
er Reilly, Stacy Tam, Donna Grant, Gregg Hetu, and Russell C. Petterpp 2009–2018
Publication Date (Web): August=
12, 2004 (Article)
Lisa C. W. Chang, Jacobien K. von Frijtag Drabbe Künzel, =
Thea Mulder-Krieger, Ronald F. Spanjersberg, Sophie F. Roerink, Gijs van=
den Hout, Margot W. Beukers, Johannes Brussee, and Adriaan P. IJzerman<=
/div>pp 2045–2053
Publication Date (Web): Sep=
tember 29, 2004 (Article)
J. Ignacio Andrés, Jes&uacut=
e;s Alcázar, José M. Alonso, Rosa M. Alvarez, Margot H. Ba=
kker, Ilse Biesmans, José M. Cid, Ana I. De Lucas, Javier Fern&aa=
cute;ndez, Luis M. Font, Koen A. Hens, Laura Iturrino, Ilse Lenaerts, So=
nia Martínez, Anton A. Megens, Joaquín Pastor, Patrick C. =
M. Vermote, and Thomas Steckler
pp 2054–2071
Publ=
ication Date (Web): November 02, 2004 (=
Article)
Jerome Guillemont, Elisabeth Pasquier, Patrice Palandjian, Dani=
el Vernier, Sandrine Gaurrand, Paul J. Lewi, Jan Heeres, Marc R. de Jong=
e, Lucien M. H. Koymans, Frits F. D. Daeyaert, Maarten H. Vinkers, Eddy =
Arnold, Kalyan Das, Rudi Pauwels, Koen Andries, Marie-Pierre de Bé=
;thune, Eva Bettens, Kurt Hertogs, Piet Wigerinck, Philip Timmerman, and=
Paul A. J. Janssen
pp 2072–2079
Publication Date=
(Web): November 18, 2004 (Article)
Antoni To=
rrens, Josep Mas, Adriana Port, José Aurelio Castrillo, Olga Sanf=
eliu, Xavier Guitart, Alberto Dordal, Gonzalo Romero, Ma Ange=
les Fisas, Elisabeth Sánchez, Enrique Hernández, Pilar P&e=
acute;rez, Raquel Pérez, and Helmut Buschmann
pp 2080–=
2092
Publication Date (Web): October 30, 2004 (Article)
Ruengwit Kitbunnadaj, Takeshi Hashimo=
to, Enzo Poli, Obbe P. Zuiderveld, Alessandro Menozzi, Ryoko Hidaka, Iwa=
n J. P. de Esch, Remko A. Bakker, Wiro M. P. B. Menge, Atsushi Yamatodan=
i, Gabriella Coruzzi, Henk Timmerman, and Rob Leurs
pp 2100–2=
107
Publication Date (Web): November 24, 2004 (Article)
Weiqin Jiang, J=
ihua Guan, Mark J. Macielag, Suying Zhang, Yuhong Qiu, Patricia Kraft, S=
heela Bhattacharjee, T. Matthew John, Donna Haynes-Johnson, Scott Lundee=
n, and Zhihua Sui
pp 2126–2133
Publication Date (=
Web): December 08, 2004 (Article)
Domi=
nique Mabire, Sophie Coupa, Christophe Adelinet, Alain Poncelet, Yvan Si=
monnet, Marc Venet, Ria Wouters, Anne S. J. Lesage, Ludy Van Beijstervel=
dt, and François Bischoff
pp 2134–2153
Pub=
lication Date (Web): January 28, 2005 (=
Article)
Eddy J. Freyne, Jean F. Lacrampe, Frederik Deroose, Gustaaf M=
. Boeckx, Marc Willems, Werner Embrechts, Erwin Coesemans, Johan J. Will=
ems, Jerome M. Fortin, Yannick Ligney, Lieve L. Dillen, Willy F. Cools, =
Jan Goossens, David Corens, Alex De Groot, and Jean P. Van Wauwe
pp=
2167–2175
Publication Date (Web): December 2=
9, 2004 (Article)
Lieven Meerpoel, L=
eo J. J. Backx, Louis J. E. Van der Veken, Jan Heeres, David Corens, Ale=
x De Groot, Frank C. Odds, Frans Van Gerven, Filip A. A. Woestenborghs, =
Andre Van Breda, Michel Oris, Pascal van Dorsselaer, Gustaaf H. M. Wille=
msens, Karen J. P. Vermuyten, Patrick J. M. G. Marichal, Hugo F. Vanden =
Bossche, Jannie Ausma, and Marcel Borgers
pp 2184–2193
Publication Date (Web): January 28, 2005 (Article)
G=
eorge V. De Lucca, Ui Tae Kim, Brian J. Vargo, John V. Duncia, Joseph B.=
Santella, III, Daniel S. Gardner, Changsheng Zheng, Ann Liauw, Zhang Wa=
ng, George Emmett, Dean A. Wacker, Patricia K. Welch, Maryanne Covington=
, Nicole C. Stowell, Eric A. Wadman, Anuk M. Das, Paul Davies, Swamy Yel=
eswaram, Danielle M. Graden, Kimberly A. Solomon, Robert C. Newton, Geor=
ge L. Trainor, Carl P. Decicco, and Soo. S. Ko
pp 2194–2211Publication Date (Web): January 14, 2005 (Article)
Iwao Ojima, Christopher P. Borella, Xinyuan Wu, Pierre-Yves Bounaud, =
Cecilia Fumero Oderda, Matthew Sturm, Michael L. Miller, Subrata Chakrav=
arty, Jin Chen, Qing Huang, Paula Pera, Tracy A. Brooks, Maria R. Baer, =
and Ralph J. Bernacki
pp 2218–2228
Publication Da=
te (Web): January 25, 2005 (Article)
Curt A=
. Dvorak, Richard Apodaca, Ann J. Barbier, Craig W. Berridge, Sandy J. W=
ilson, Jamin D. Boggs, Wei Xiao, Timothy W. Lovenberg, and Nicholas I. C=
arruthers
pp 2229–2238
Publication Date (Web): =
strong>February 05, 2005 (Article)
<=
div class=3D"DOI">DOI: 10.1021/jm049212n
Abstract | <=
a class=3D"articleLink" href=3D"/doi/suppl/10.1021/jm049212n">Supporting=
Info
Wil=
liam J. Hoekstra, Hari S. Patel, Xi Liang, Jean-Baptiste E. Blanc, Denni=
s O. Heyer, Timothy M. Willson, Marie A. Iannone, Sue H. Kadwell, Lisa A=
. Miller, Kenneth H. Pearce, Catherine A. Simmons, and Jean Shearin
pp 2243–2247
Publication Date (Web): Decembe=
r 13, 2004 (Brief Article)
Pratik V. Devasthale, Sean Chen, Yoon=
Jeon, Fucheng Qu, Chunning Shao, Wei Wang, Hao Zhang, Michael Cap, Denn=
is Farrelly, Rajasree Golla, Gary Grover, Thomas Harrity, Zhengping Ma, =
Lisa Moore, Jimmy Ren, Ramakrishna Seethala, Lin Cheng, Paul Sleph, Wei =
Sun, Aaron Tieman, John R. Wetterau, Arthur Doweyko, Gamini Chandrasena,=
Shu Y. Chang, W. Griffith Humphreys, Vito G. Sasseville, Scott A. Bille=
r, Denis E. Ryono, Fred Selan, Narayanan Hariharan, and Peter T. W. Chen=
g
pp 2248–2250
Publication Date (Web): N=
ovember 13, 2004 (Brief Article)
To jump to an article, select a journal and fill =
in volume and article's first page or specify the DOI of the article=
in the DOI box, and then click "Go".=
div>